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(2R,3S)-Azelaprag

SKU: orb1745251

Description

This compound is a potent apelin receptor agonist with an EC50 of 12 nM. It serves as a valuable research tool for investigating cardiovascular and metabolic diseases, including heart failure, diabetes, and hypertension, in both in vitro and in vivo models.

Research Area

Pharmacology & Drug Discovery

Images & Validation

Key Properties

CAS Number2049979-31-7
MW523.61
Purity99.35%
FormulaC25H29N7O4S
SMILESN(S([C@@H]([C@@H](C)C=1N=CC(C)=CN1)C)(=O)=O)C=2N(C(=NN2)C=3C=C(C)C=NC3)C4=C(OC)C=CC=C4OC
TargetApelin receptor

Bioactivity

Target IC50
Apelin receptor:0.012 µM

Storage & Handling

StoragePowder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.
Expiration Date12 months from date of receipt.
DisclaimerFor research use only

Alternative Names

(2R,3S)N(4(2,6dimethoxyphenyl)5(5methylpyridin3yl)4H1,2,4triazol3yl)3(5methylpyrimidin2yl)butane2sulfonamide, Azelaprag, Apelinreceptor, Apelin receptor
Quality Guarantee

Quality Guarantee

Explore bioreagents carefree to elevate your research. All our products are rigorously tested for performance. If a product does not perform as described on its datasheet, our scientific support team will provide expert troubleshooting, a prompt replacement, or a refund. For full details, please see our Terms & Conditions and Buying Guide. Contact us at [email protected].

Key Properties

No computed properties available.

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Protocol Information

(2R,3S)-Azelaprag (orb1745251)

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(Recommended: An additional animal making an allowance for loss during the experiment)

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Available Sizes

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1 mg
¥ 3,120.00
5 mg
¥ 7,280.00
1 ml x 10 mM (in DMSO)
¥ 8,190.00
10 mg
¥ 11,830.00
25 mg
¥ 24,310.00
50 mg
¥ 38,610.00
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