Atopaxar Hydrobromide

SKU: orb1705932

Description

Atopaxar is a reversible antagonist of the PAR-1 thrombin receptor, inhibiting platelet activation pathways. It has been studied in preclinical and clinical research contexts for the potential management of coronary artery disease and acute coronary syndromes.

Research Area

Cardiovascular Research, Cell Biology, Epigenetics & Chromatin, Pharmacology & Drug Discovery, Signal Transduction, Stem Cell & Developmental Biology

Images & Validation

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Key Properties

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CAS Number	474550-69-1
MW	608.54
Purity	100.00%
Formula	C₂₉H₃₉BrFN₃O₅
SMILES	Br.CCOc1cc2CN(CC(=O)c3cc(N4CCOCC4)c(OC)c(c3)C(C)(C)C)C(=N)c2c(F)c1OCC
Target	Protease-activated Receptor,Apoptosis,JAK
Solubility	DMSO:10 mM

Bioactivity

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Target IC50	PAR1:5.1 nM

Storage & Handling

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Storage	Powder: -20°C for 3 years \| In solvent: -80°C for 1 year \| Shipping with blue ice/Shipping at ambient temperature.
Expiration Date	12 months from date of receipt.
Disclaimer	For research use only

Alternative Names

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E5555, E-5555, E 5555, atherothrombotic, Atopaxar, Atopaxar Hydrobromide, PAR-1, platelets, inhibit, Inhibitor, ER 172594-06, Thrombin receptors, thrombin, receptor, receptor-1, signaling, Protease Activated Receptor (PAR), ProteaseactivatedReceptor, protease-activated, Proteaseactivated Receptor

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Compound Identifiers

PubChem CID

22929978 ↗

Key Properties

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No computed properties available.

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