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BI-2081

SKU: orb1744175

Description

BI-2081 is a potent and selective partial agonist of the GPR40 (FFAR1) receptor with an EC50 of 4 nM. It stimulates insulin secretion in a glucose-dependent manner and has demonstrated efficacy in reducing blood glucose levels in preclinical models of type 2 diabetes, making it a valuable tool for metabolic disease research.

Research Area

Metabolism Research, Pharmacology & Drug Discovery

Images & Validation

Key Properties

CAS Number1458656-71-7
MW534.62
FormulaC32H35FO6
SMILESO([C@H]1C=2C(=C(C=CC2F)C3=C(C)C=C(OCCC(C)(C)O)C=C3C)CC1)C=4C=C5C(=CC4)[C@H](CC(O)=O)CO5
TargetGPCR,Others

Storage & Handling

Storage-20°C
Expiration Date12 months from date of receipt.
DisclaimerFor research use only
Quality Guarantee

Quality Guarantee

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Key Properties

No computed properties available.

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Protocol Information

BI-2081 (orb1744175)

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