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BRD2879

SKU: orb1700963

Description

BRD2879 is a potent, cell-permeable small molecule inhibitor targeting the IDH1-R132H mutant protein with an IC50 of 50 nM. It is a valuable research tool for studying oncogenic metabolism in vitro and has shown utility in preclinical models for investigating gliomas and other cancers harboring this mutation.

Research Area

Metabolism Research

Images & Validation

Key Properties

CAS Number1304750-47-7
MW571.70
FormulaC30H38FN3O5S
SMILESO=S1(=O)C=2C(O[C@@H](CN(C(NC3CCCCC3)=O)C)[C@H](C)CN1[C@H](CO)C)=CC(C#CC4=CC(F)=CC=C4)=CC2
TargetOthers,Isocitrate Dehydrogenase (IDH)

Storage & Handling

Storage-20°C
Expiration Date12 months from date of receipt.
DisclaimerFor research use only
Quality Guarantee

Quality Guarantee

Explore bioreagents carefree to elevate your research. All our products are rigorously tested for performance. If a product does not perform as described on its datasheet, our scientific support team will provide expert troubleshooting, a prompt replacement, or a refund. For full details, please see our Terms & Conditions and Buying Guide. Contact us at [email protected].

Key Properties

No computed properties available.

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Protocol Information

BRD2879 (orb1700963)

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