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CYT-1010

SKU: orb1709949

Description

CYT-1010 is a potent and selective mu-opioid receptor agonist, demonstrating high functional bias with an EC50 of 0.0053 nM for inhibiting cAMP production versus 13.1 nM for β-arrestin recruitment. This profile makes it a valuable research tool for investigating biased agonism, G-protein signaling pathways, and pain-related in vitro and in vivo studies.

Research Area

Metabolism Research, Neuroscience, Pharmacology & Drug Discovery

Images & Validation

Key Properties

CAS Number213769-33-6
MW624.73
FormulaC35H40N6O5
SMILESC(C=1C=2C(NC1)=CC=CC2)[C@H]3C(=O)N[C@@H](CC4=CC=CC=C4)C(=O)NCCCC[C@@H](NC([C@H](CC5=CC=C(O)C=C5)N)=O)C(=O)N3
TargetOthers,Opioid Receptor

Storage & Handling

Storage-20°C
Expiration Date12 months from date of receipt.
DisclaimerFor research use only

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Key Properties

No computed properties available.

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CYT-1010 (orb1709949)

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