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DPP-4/GPR119 modulator 1

SKU: orb1982858

Description

DPP-4/GPR119 modulator 1 (Compound 22) is an orally bioavailable dual-acting agent, functioning as a DPP-IV inhibitor and a GPR119 agonist. It lowers blood glucose in vivo and shows moderate hERG channel inhibition (IC50 = 4.9 µM), making it a useful tool for investigating diabetes and metabolic disease pathways.

Research Area

Metabolism Research, Pharmacology & Drug Discovery, Protein Biochemistry

Images & Validation

Key Properties

CAS Number2411099-68-6
MW623.15
FormulaC30H39ClN10O3
SMILESCl.CC#CCn1c(nc2n(C)c(=O)n(CCCN3CCN(CC3)c3nc(no3)-c3ccccc3)c(=O)c12)N1CCC[C@@H](N)C1
TargetOthers,Proteasome,GPCR,Potassium Channel

Storage & Handling

Storage-20°C
Expiration Date12 months from date of receipt.
DisclaimerFor research use only
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Key Properties

No computed properties available.

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Protocol Information

DPP-4/GPR119 modulator 1 (orb1982858)

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