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Fedovapagon

SKU: orb1707315

Description

Fedovapagon (VA106483) is a selective and potent vasopressin V2 receptor agonist. It is utilized in research models, such as zebrafish for studying angiogenesis, and in investigations of urological conditions including overactive bladder and nocturia.

Research Area

Pharmacology & Drug Discovery

Images & Validation

Key Properties

CAS Number347887-36-9
MW462.58
Purity99.46%
FormulaC27H34N4O3
SMILES[H][C@]1(CCCN1C(=O)NCc1ccc(cc1C)C(=O)N1CCCCc2ccccc12)C(=O)N(C)C
TargetVasopressin Receptor
Solubility10% DMSO+40% PEG300+5% Tween 80+45% Saline:2 mg/mL (4.32 mM);DMSO:50 mg/mL (108.09 mM)

Bioactivity

Target IC50
V2 receptor:24 nM (EC50)
In Vivo
In rats, oral administration of fedovapagon at a dose of 1 mg/kg results in an 81% inhibition rate of urine output.

Storage & Handling

StoragePowder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.
Expiration Date12 months from date of receipt.
DisclaimerFor research use only

Alternative Names

A106483, VasopressinReceptor, Vasopressin Receptor, Vasopressin receptor 2, V2R, VA483
Quality Guarantee

Quality Guarantee

Explore bioreagents carefree to elevate your research. All our products are rigorously tested for performance. If a product does not perform as described on its datasheet, our scientific support team will provide expert troubleshooting, a prompt replacement, or a refund. For full details, please see our Terms & Conditions and Buying Guide. Contact us at [email protected].

Key Properties

No computed properties available.

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Protocol Information

Fedovapagon (orb1707315)

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Step 1: Enter information below

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% DMSO +
%+
% Tween 80 +
%

Available Sizes

Select a size below

5 mg
¥ 2,080.00
1 ml x 10 mM (in DMSO)
¥ 2,210.00
10 mg
¥ 2,860.00
25 mg
¥ 5,720.00
50 mg
¥ 9,490.00
100 mg
¥ 13,260.00
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