Queen's Award Received in 2021 ISO 9001 Certified Delivered over 1,000,000 bio-reagents to life science researchers Trusted by Life Science Communities
Cart summary

You have no items in your shopping cart.

Fluorobexarotene

SKU: orb1709684

Description

Fluorobexarotene is a potent RXRα agonist with a Ki of 12 nM and an EC50 of 43 nM, exhibiting 75% greater binding affinity than Bexarotene. This small molecule is a valuable research tool for studying RXR-mediated pathways in oncology and metabolic diseases, applicable in both in vitro and in vivo experimental models.

Research Area

Metabolism Research

Images & Validation

Key Properties

CAS Number1190848-23-7
MW366.47
Purity99.08% (May vary between batches)
FormulaC24H27FO2
SMILESCC1=CC2=C(C=C1C(=C)C1=CC(F)=C(C=C1)C(O)=O)C(C)(C)CCC2(C)C
TargetRetinoid Receptor
SolubilityDMSO:5 mg/mL (13.64 mM)

Bioactivity

Target IC50
RXRα:12 nM (Ki)|RXRα:43 nM (EC50)

Storage & Handling

Storage-20°C
Expiration Date12 months from date of receipt.
DisclaimerFor research use only

Alternative Names

RXRα, Retinoid Receptor, RetinoidReceptor, Fluorobexarotene
Quality Guarantee

Quality Guarantee

Explore bioreagents carefree to elevate your research. All our products are rigorously tested for performance. If a product does not perform as described on its datasheet, our scientific support team will provide expert troubleshooting, a prompt replacement, or a refund. For full details, please see our Terms & Conditions and Buying Guide. Contact us at [email protected].

Key Properties

No computed properties available.

Protocol Information

Available Sizes

Select a size below

1 mg
$ 230.00
1 ml x 10 mM (in DMSO)
$ 420.00
5 mg
$ 510.00
10 mg
$ 730.00
25 mg
$ 1,110.00
50 mg
$ 1,490.00
100 mg
$ 1,990.00
500 mg
$ 3,930.00
DispatchUsually dispatched within 3-5 working days
Bulk Enquiry