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GAT100

SKU: orb1739179

Description

GAT-100 is a covalent negative allosteric modulator (NAM) of CB1R that paradoxically enhances orthosteric agonist binding. This unique covalent probe is a valuable tool for mapping allosteric sites and investigating CB1 receptor modulation in both in vitro binding assays and cellular signaling studies.

Images & Validation

Key Properties

CAS Number1663564-42-8
MW432.58
FormulaC25H28N4OS
SMILESC(C)C=1C=2C(NC1C(NCCC3=CC=C(C=C3)N4CCCCC4)=O)=CC=C(N=C=S)C2
TargetOthers

Storage & Handling

Storage-20°C
Expiration Date12 months from date of receipt.
DisclaimerFor research use only
Quality Guarantee

Quality Guarantee

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Key Properties

No computed properties available.

Protocol Information

Available Sizes

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25 mg
$ 1,860.00
50 mg
$ 2,420.00
100 mg
$ 3,140.00
DispatchUsually dispatched within 8-10 weeks
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