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GPR81 agonist 2

SKU: orb1744676

Description

GPR81 agonist 2 is a potent small molecule activator of the GPR81 receptor, with EC50 values of 0.023 µM (hGPR81) and 0.123 µM (hGPR109A). It serves as a valuable research tool for studying lactate signaling in metabolic disorders, inflammation, and cancer within in vitro and in vivo experimental models.

Research Area

Metabolism Research, Pharmacology & Drug Discovery

Images & Validation

Key Properties

CAS Number1143024-28-5
MW603.11
FormulaC26H27ClN6O5S2
SMILESS(=O)(=O)(C=1C=C2C(N=C(NC(NC(=O)C3=CC(=C(OCC)C=C3Cl)N4C=CC=N4)=O)S2)=CC1)C5CCN(C)CC5
TargetGPCR,Others,HCAR

Storage & Handling

Storage-20°C
Expiration Date12 months from date of receipt.
DisclaimerFor research use only
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Quality Guarantee

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Key Properties

No computed properties available.

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Protocol Information

GPR81 agonist 2 (orb1744676)

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(Recommended: An additional animal making an allowance for loss during the experiment)

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