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GR103545

SKU: orb1298083

Description

GR103545 is a selective κ-opioid receptor (KOR) agonist widely employed as a radiotracer for positron emission tomography (PET) imaging. It enables the in vivo visualization and quantification of KOR distribution and occupancy in neurological and psychiatric research.

Research Area

Metabolism Research, Neuroscience, Pharmacology & Drug Discovery

Images & Validation

Key Properties

CAS Number126766-43-6
MW530.4
Purity97.19% (May vary between batches)
FormulaC23H29Cl2N3O7
SMILESOC(=O)\C=C\C(O)=O.COC(=O)N1CCN([C@H](CN2CCCC2)C1)C(=O)Cc1ccc(Cl)c(Cl)c1
TargetOthers,Opioid Receptor
SolubilityDMSO:60 mg/mL (113.12 mM);10% DMSO+40% PEG300+5% Tween 80+45% Saline:2 mg/mL (3.77 mM)

Storage & Handling

Storage-20°C
Expiration Date12 months from date of receipt.
DisclaimerFor research use only

Alternative Names

κ-opioid receptor, κ-OR, GR 103545, GR103545, GR-103545, Opioid Receptor, inhibit, Inhibitor, imaging
Quality Guarantee

Quality Guarantee

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Key Properties

No computed properties available.

Protocol Information

Available Sizes

Select a size below

1 mg
$ 130.00
2 mg
$ 190.00
5 mg
$ 240.00
1 ml x 10 mM (in DMSO)
$ 310.00
10 mg
$ 340.00
25 mg
$ 580.00
50 mg
$ 810.00
100 mg
$ 1,110.00
DispatchUsually dispatched within 3-5 working days
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