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IC87201

SKU: orb1299890

Description

IC87201 is a selective small-molecule inhibitor targeting the PDZ domains of nNOS and PSD-95. It has demonstrated significant potential in preclinical research, showing efficacy in cellular assays and animal models for conditions such as ischemic stroke and pain modulation.

Research Area

Neuroscience, Pharmacology & Drug Discovery

Images & Validation

Key Properties

CAS Number866927-10-8
MW309.15
Purity97.44%
FormulaC13H10Cl2N4O
SMILESOc1c(Cl)cc(Cl)cc1CNc1ccc2nn[nH]c2c1
TargetiGluR
SolubilityDMSO:28 mg/mL (90.57 mM)

Bioactivity

In Vitro
IC87201 have been presented as efficient inhibitors of the nNOS/PSD-95 protein-protein interaction and shown great promise in cellular experiments and animal models of ischemic stroke and pain. Under the applied in vitro conditions.

Storage & Handling

StoragePowder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.
Expiration Date12 months from date of receipt.
DisclaimerFor research use only

Alternative Names

Inhibitor, IC87201, IC-87201, IC 87201, iGluR, nNOS-PDZ/PSD-95-PDZ, Ionotropic glutamate receptors, inhibit
Quality Guarantee

Quality Guarantee

Explore bioreagents carefree to elevate your research. All our products are rigorously tested for performance. If a product does not perform as described on its datasheet, our scientific support team will provide expert troubleshooting, a prompt replacement, or a refund. For full details, please see our Terms & Conditions and Buying Guide. Contact us at [email protected].

Key Properties

No computed properties available.

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IC87201 (orb1299890)

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1 ml x 10 mM (in DMSO)
¥ 910.00
25 mg
¥ 1,170.00
50 mg
¥ 1,690.00
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