Cart summary

You have no items in your shopping cart.

NH2-c[X-R-L-S-X]-K-G-P-(D-2Nal)

SKU: orb1981233

Description

This macrocyclic APJ receptor agonist, an analogue of Ape13, exhibits potent binding affinity (Ki = 5.7 nM) with Gα12-biased signaling and an improved pharmacokinetic profile. It is a valuable research tool for studying apelin receptor function in cardiovascular and metabolic diseases, suitable for both in vitro signaling studies and in vivo physiological research.

Research Area

Pharmacology & Drug Discovery

Images & Validation

Key Properties

CAS Number2891469-81-9
MW1020.18
FormulaC49H73N13O11
TargetApelin receptor,Others

Storage & Handling

Storage-20°C
Expiration Date12 months from date of receipt.
DisclaimerFor research use only
Quality Guarantee

Quality Guarantee

Explore bioreagents carefree to elevate your research. All our products are rigorously tested for performance. If a product does not perform as described on its datasheet, our scientific support team will provide expert troubleshooting, a prompt replacement, or a refund. For full details, please see our Terms & Conditions and Buying Guide. Contact us at [email protected].

Documents Download

Datasheet
Product Information
Download

Request a Document

Protocol Information

NH2-c[X-R-L-S-X]-K-G-P-(D-2Nal) (orb1981233)

  • Star
  • Star
  • Star
  • Star
  • Star
  • 0.0
Based on 0 reviews

Participating in our Biorbyt product reviews program enables you to support fellow scientists by sharing your firsthand experience with our products.

Login to Submit a Review

No reviews yet

Step 1: Enter information below

(Recommended: An additional animal making an allowance for loss during the experiment)

Step 2: Enter the in vivo formulation

(This is only the calculator, not formulation. Please contact us first if there is no in vivo formulation at the solubility Section.)

% DMSO +
%+
% Tween 80 +
%