Opioid receptor agonist 1

SKU: orb2944935

Description

Compound 2638-28 is a potent, orally bioavailable pan-opioid receptor agonist with high affinity for MOR (Ki=5 nM), DOR (Ki=24 nM), and KOR (Ki=212 nM). It demonstrates significant analgesic efficacy in validated in vivo models, including the mouse tail-flick and acetic acid writhing tests, making it a useful research tool for studying pain mechanisms and opioid receptor pharmacology.

Research Area

Metabolism Research, Neuroscience, Pharmacology & Drug Discovery

Images & Validation

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Key Properties

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MW	515.73
Formula	C₃₂H₄₅N₅O
Target	Opioid Receptor

Storage & Handling

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Storage	-20°C
Expiration Date	12 months from date of receipt.
Disclaimer	For research use only

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Gene Symbol

Opioid Receptor

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