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Otenabant

SKU: orb1224245

Description

A potent, and selective CB1 receptor antagonist with Ki of 0.7 nM/0.12 nM in binding and functional assays respectively; has low affinity (Ki=7600 nM) for human CB2 receptors; reverses cannabinoid agonist mediated responses, reduces food intake, and increases energy expenditure and fat oxidation in rodents.ObesityPhase 3 Discontinued

Images & Validation

Key Properties

CAS Number686344-29-6
MW510.4
Purity>98% (HPLC)
FormulaC25H25Cl2N7O
TargetCB1

Storage & Handling

StorageStorage temperature: -20°C. Stability: ≥ 2 years
DisclaimerFor research use only

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Otenabant (orb1224245)

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% DMSO +
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Available Sizes

Select a size below

100 mg
200 mg
500 mg
2 mg
¥ 1,040.00
5 mg
¥ 1,690.00
10 mg
¥ 1,950.00
25 mg
¥ 3,510.00
50 mg
¥ 5,980.00