P2Y2R/GPR17 antagonist 1

SKU: orb1687624

Description

Compound 14m is a dual antagonist targeting both the P2Y2 and GPR17 receptors, exhibiting IC50 values of 3.17 µM and 1.67 µM, respectively. This small molecule is a valuable research tool for investigating purinergic signaling in models of inflammation, neuropathic pain, and demyelinating diseases in vitro.

Research Area

Metabolism Research, Neuroscience, Pharmacology & Drug Discovery

Images & Validation

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Key Properties

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CAS Number	2395016-49-4
MW	432.83
Purity	98.21% (May vary between batches)
Formula	C₁₉H₁₃ClN₂O₆S
SMILES	[O-][N+](=O)c1cccc(OS(=O)(=O)c2ccc(NC(=O)c3ccccc3Cl)cc2)c1
Target	P2Y Receptor,GPCR
Solubility	DMSO:112.5 mg/mL (259.92 mM)

Storage & Handling

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Storage	-20°C
Expiration Date	12 months from date of receipt.
Disclaimer	For research use only

Alternative Names

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GPR17

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Compound Identifiers

PubChem CID

162646428 ↗

Key Properties

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No computed properties available.

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