RXFP1 receptor agonist-3

SKU: orb1943520

Description

Example 223 is a potent small molecule agonist of the human RXFP1 receptor with an EC₅₀ of 2 nM, demonstrated to inhibit cAMP production in HEK293 cells. This tool compound is valuable for in vitro studies investigating relaxin signaling pathways and receptor pharmacology in cardiovascular and fibrotic disease research.

Research Area

Pharmacology & Drug Discovery

Images & Validation

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Key Properties

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CAS Number	2924767-53-1
MW	831.72
Formula	C₄₂H₃₄F₉N₃O₅
SMILES	C(=C/1\[C@@]2([C@@H](NC(=O)C3=CC(=CC=C3OC)C4=CC(C(OC(NC5=C(F)C=CC=C5)=O)C(F)(F)F)=CC=C4F)[C@@H](C(NC6=CC(C(F)(F)F)=C(F)C=C6)=O)[C@]1(CC2)[H])[H])\C7CC7
Target	RXFP receptor,Others

Storage & Handling

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Storage	-20°C
Expiration Date	12 months from date of receipt.
Disclaimer	For research use only

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Compound Identifiers

PubChem CID

171361115 ↗

Key Properties

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No computed properties available.

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