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RXFP1 receptor agonist-3

SKU: orb1943520

Description

Example 223 is a potent small molecule agonist of the human RXFP1 receptor with an EC₅₀ of 2 nM, demonstrated to inhibit cAMP production in HEK293 cells. This tool compound is valuable for in vitro studies investigating relaxin signaling pathways and receptor pharmacology in cardiovascular and fibrotic disease research.

Research Area

Pharmacology & Drug Discovery

Images & Validation

Key Properties

CAS Number2924767-53-1
MW831.72
FormulaC42H34F9N3O5
SMILESC(=C/1\[C@@]2([C@@H](NC(=O)C3=CC(=CC=C3OC)C4=CC(C(OC(NC5=C(F)C=CC=C5)=O)C(F)(F)F)=CC=C4F)[C@@H](C(NC6=CC(C(F)(F)F)=C(F)C=C6)=O)[C@]1(CC2)[H])[H])\C7CC7
TargetOthers,RXFP receptor

Storage & Handling

Storage-20°C
Expiration Date12 months from date of receipt.
DisclaimerFor research use only
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Key Properties

No computed properties available.

Protocol Information