CB2 receptor agonist 2

SKU: orb1306124

Description

Research Area

Pharmacology & Drug Discovery

Images & Validation

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Key Properties

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CAS Number	1314230-75-5
MW	488.62
Purity	99.75%
Formula	C₃₀H₃₆N₂O₄
SMILES	N(C(=O)C=1C(=O)C=2C(N(CCCCC)C1)=C(OC)C=C(C2)C3=CC=CO3)C45CC6CC(C4)CC(C5)C6
Target	Cannabinoid Receptor
Solubility	DMSO:3 mg/mL (6.14 mM)

Bioactivity

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Target IC50	CB2:8.5 nM (Ki)
In Vivo	CB2 receptor agonist 2 (compound 4g) (1 and 3 mg/kg; 1 hour) is highly potent, showing maximal effect at 1 mg/kg, with antihyperalgesic effects that are effective in the first phase of the nocifensive response and are strongly reduced by AM630, a CB2-selective antagonist/inverse agonist . Read more...
In Vitro	CB2 receptor agonist 2 (compound 4g) (1 μM, 72 hours) exhibits minimal to no cytotoxicity in Hep-G2 cells.

Storage & Handling

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Storage	Powder: -20°C for 3 years \| In solvent: -80°C for 1 year \| Shipping with blue ice/Shipping at ambient temperature.
Expiration Date	12 months from date of receipt.
Disclaimer	For research use only

Alternative Names

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CB2R, CB2 receptor agonist 2, CannabinoidReceptor, Cannabinoid Receptor, 4-Quinolone-3-Carboxamide Furan CB2 Agonist, ZINC 72105556, ZINC72105556, ZINC-72105556

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Compound Identifiers

PubChem CID

53387350 ↗

Key Properties

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No computed properties available.

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