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GSK0660

SKU: orb1305182

Description

GSK0660 is a potent and selective PPARβ/δ antagonist with inverse agonist properties. This small molecule inhibitor is widely used in metabolic, inflammatory, and cancer research, facilitating both in vitro mechanistic studies and in vivo model investigations.

Research Area

Metabolism Research, Molecular Biology

Images & Validation

Key Properties

CAS Number1014691-61-2
MW418.49
Purity99.71%
FormulaC19H18N2O5S2
SMILESS(NC1=C(OC)C=C(NC2=CC=CC=C2)C=C1)(=O)(=O)C3=C(C(OC)=O)SC=C3
TargetPPAR
SolubilityEthanol:4.19 mg/mL (10.01 mM);10% DMSO+40% PEG300+5% Tween 80+45% Saline:2 mg/mL (4.78 mM);DMSO:117.5 mg/mL (280.77 mM)

Bioactivity

Target IC50
PPARβ/δ:155 nM

Storage & Handling

StoragePowder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.
Expiration Date12 months from date of receipt.
DisclaimerFor research use only

Alternative Names

inhibit, GSK0660, GSK-0660, GSK 0660, Inhibitor, PPARδ, PPARβ, PPAR, Peroxisome proliferator-activated receptors

Similar Products

  • GSK0660 [orb1223455]

    >98% (HPLC)

    1014691-61-2

    418.5

    C19H18N2O5S2

    2 mg, 5 mg, 10 mg, 25 mg, 50 mg, 100 mg, 500 mg, 1 g
Quality Guarantee

Quality Guarantee

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Key Properties

No computed properties available.

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Protocol Information

GSK0660 (orb1305182)

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% DMSO +
%+
% Tween 80 +
%

Available Sizes

Select a size below

2 mg
¥ 1,040.00
1 ml x 10 mM (in DMSO)
¥ 1,430.00
5 mg
¥ 1,430.00
10 mg
¥ 1,950.00
25 mg
¥ 3,120.00
50 mg
¥ 5,590.00
100 mg
¥ 8,060.00
500 mg
¥ 16,900.00
DispatchUsually dispatched within 3-5 working days
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