Lys-[Des-Arg9]Bradykinin TFA

SKU: orb1983569

Description

Lys-[Des-Arg9]Bradykinin TFA is a naturally occurring kinin that serves as a potent and highly selective agonist for the bradykinin B1 receptor, demonstrating binding affinities (K i values) of 0.12 nM, 1.7 nM, and 0.23 nM for the human, mouse, and rabbit B1 receptors, respectively. This compound exhibits low inhibitory activity on B2 receptors.

Research Area

Pharmacology & Drug Discovery

Images & Validation

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Key Properties

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CAS Number	2763588-90-3
MW	1260.24
Formula	C₅₄H₇₅F₆N₁₃O₁₅
SMILES	OC(C(F)(F)F)=O.O=C(N1[C@@H](CCC1)C(NCC(N[C@H](C(N[C@@H](CO)C(N2[C@@H](CCC2)C(N[C@H](C(O)=O)CC3=CC=CC=C3)=O)=O)=O)CC4=CC=CC=C4)=O)=O)[C@H]5N(CCC5)C([C@H](CCCNC(N)=N)NC([C@@H](N)CCCCN)=O)=O.OC(C(F)(F)F)=O
Target	Bradykinin Receptor

Storage & Handling

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Storage	-20°C
Disclaimer	For research use only

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Compound Identifiers

PubChem CID

163342333 ↗

Key Properties

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No computed properties available.

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