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(-)-OPC-51803

SKU: orb1745241

Description

(-)-OPC-51803 is a selective vasopressin V2 receptor agonist utilized in pharmacological research. It serves as a key tool compound for investigating renal water reabsorption mechanisms in vitro and evaluating potential therapies for conditions like nocturia in vivo models.

Research Area

Metabolism Research, Neuroscience

Images & Validation

Key Properties

CAS Number192514-57-1
MW454
Purity99.59%
FormulaC26H32ClN3O2
SMILESC(=O)(N1C=2C([C@H](CC(NC(C)C)=O)CCC1)=CC=CC2)C3=C(Cl)C=C(C=C3)N4CCCC4
TargetEndogenous Metabolite,AChR
SolubilityDMSO:45 mg/mL (99.12 mM);10% DMSO+40% PEG300+5% Tween-80+45% Saline:2 mg/mL (4.41 mM)

Bioactivity

Target IC50
V2 receptor:0.39 µM|V2 receptor:0.98 µM

Storage & Handling

StoragePowder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.
Expiration Date12 months from date of receipt.
DisclaimerFor research use only

Alternative Names

OPC51803, OPC-51803, OPC 51803, ADH, (S)2(1(2chloro4(pyrrolidin1yl)benzoyl)2,3,4,5tetrahydro1Hbenzo[b]azepin5yl)Nisopropylacetamide(192514548Freebase)

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Quality Guarantee

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Key Properties

No computed properties available.

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Protocol Information

(-)-OPC-51803 (orb1745241)

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% DMSO +
%+
% Tween 80 +
%

Available Sizes

Select a size below

1 mg
¥ 2,080.00
5 mg
¥ 3,900.00
10 mg
¥ 5,590.00
25 mg
¥ 8,320.00
50 mg
¥ 11,180.00
100 mg
¥ 14,690.00
200 mg
¥ 19,760.00
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