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PSB-KD477

SKU: orb1739868

Description

PSB-KD477 is a potent and selective synthetic agonist for the orphan receptor GPR18, demonstrating superior activity to THC in β-arrestin recruitment assays without activating CB1, CB2, or GPR55. Its distinct indole-based structure makes it a valuable chemical probe for validating GPR18's physiological roles in vitro and for exploring its involvement in immune regulation and cancer biology, as suggested by preliminary research.

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Key Properties

CAS Number2488763-19-3
MW392.45
FormulaC21H24N6O2
SMILESO=C1C=2N3C(=NC2N(C)C(=O)N1C)N(CCC=4C=5C(NC4)=CC=CC5)CCCC3
TargetOthers

Storage & Handling

Storage-20°C
Expiration Date12 months from date of receipt.
DisclaimerFor research use only

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Key Properties

No computed properties available.

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PSB-KD477 (orb1739868)

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