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TGR5 Receptor Agonist 4

SKU: orb1943763

Description

TGR5 Receptor Agonist 4 is a potent and selective small molecule agonist for the bile acid receptor TGR5, demonstrating EC50 values of 2 nM (hTGR5) and 3 nM (mTGR5). It is a valuable research tool for studying TGR5-mediated metabolic functions, including glucose homeostasis and body weight regulation, in both in vitro and in vivo models.

Research Area

Pharmacology & Drug Discovery

Images & Validation

Key Properties

CAS Number1872436-42-4
MW470.95
FormulaC25H27ClN2O5
SMILESC(OCC1=C(OC)C=CC=C1)(=O)C=2[C@@H](CC(=O)N(C[C@H]3CCCO3)C2C)C=4C=CC(Cl)=NC4
TargetOthers,GPCR19

Storage & Handling

Storage-20°C
Expiration Date12 months from date of receipt.
DisclaimerFor research use only

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Quality Guarantee

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Key Properties

No computed properties available.

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TGR5 Receptor Agonist 4 (orb1943763)

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Step 1: Enter information below

(Recommended: An additional animal making an allowance for loss during the experiment)

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