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Tofacitinib

SKU: orb1224990

Description

Tofacitinib (CP-690550) is a potent, specific, orally active inhibitor of JAK3 with IC50 of 1 nM in cell-free assays; displays 20- to 100-fold less potency for JAK2 and JAK1 (IC50=20 nM and 112 nM, respectively).

Images & Validation

Key Properties

CAS Number477600-75-2
MW312.4
Purity>98% (HPLC)
FormulaC16H20N6O
TargetJAK1|JAK2|JAK3|Lck|ROCK2

Storage & Handling

StorageStorage temperature: -20°C. Stability: ≥ 2 years
Expiration Date12 months from date of receipt.
DisclaimerFor research use only

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Tofacitinib (orb1224990)

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% DMSO +
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% Tween 80 +
%

Available Sizes

Select a size below

5 mg
¥ 910.00
10 mg
¥ 1,170.00
25 mg
¥ 1,300.00
50 mg
¥ 1,560.00
100 mg
¥ 1,950.00
200 mg
¥ 2,600.00
500 mg
¥ 4,550.00