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GPR40 agonist 5

SKU: orb1687502

Description

GPR40 agonist 5 is a potent and orally active agonist of GPR40 (EC50 = 47 nM). It effectively lowers blood glucose and improves glucose tolerance in preclinical models, demonstrating utility for in vivo research on type 2 diabetes and in vitro studies of FFAR1 signaling pathways.

Research Area

Metabolism Research, Pharmacology & Drug Discovery

Images & Validation

Key Properties

CAS Number2443384-60-7
MW440.49
FormulaC27H24N2O4
SMILESC(OC1=CC=C(C(CC(O)=O)C#CC)C=C1)C2=CN3C(=NC(=C3)C4=CC=C(OC)C=C4)C=C2
TargetOthers,GPCR

Storage & Handling

Storage-20°C
Expiration Date12 months from date of receipt.
DisclaimerFor research use only

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Key Properties

No computed properties available.

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Protocol Information

GPR40 agonist 5 (orb1687502)

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Step 1: Enter information below

(Recommended: An additional animal making an allowance for loss during the experiment)

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