PAR4 antagonist 3

SKU: orb3134153

Description

PAR4 antagonist3 (Compound 36) is a selective antagonist of protease-activated receptor 4 (PAR4). It exhibits antiplatelet activity with an IC50 of 26.1 nM and enhances metabolic stability in human liver microsomes, with a half-life (T1/2) of 97.6 minutes.

Research Area

Pharmacology & Drug Discovery

Images & Validation

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Key Properties

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CAS Number	3057206-40-0
MW	453.44
Formula	C₂₂H₁₆FN₃O₅S
SMILES	FC1=CC=C(OCC2OC3=C(OC2)C=CC=4C=C(OC34)C=5N=C6SC(=NN6C5)OC)C=C1
Target	Protease-activated Receptor

Storage & Handling

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Storage	-20°C
Expiration Date	12 months from date of receipt.
Disclaimer	For research use only

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Gene Symbol

Protease-activated Receptor

Protocol Information

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Purity:	> 95% by hplc
MW:	1409.72 Da
Structure:	Pal-Ser-Gly-Arg-Arg-Tyr-Gly-His-Ala-Leu-Arg-NH2

CAS Number:	3024653-17-3
MW:	371.84
Formula:	C₁₈H₁₄ClN₃O₂S

CAS Number:	13198-99-7
MW:	298.29
Formula:	C₁₇H₁₄O₅

CAS Number:	170632-41-4
MW:	356.42
Formula:	C₂₃H₂₀N₂O₂

PAR4 antagonist 3

Description

Research Area

Images & Validation

Key Properties

Storage & Handling

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